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Bornyl derivatives of p-(Benzyloxy)phenylpropionic acid: In vivo evaluation of antidiabetic activity
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Bornyl derivatives of p-(Benzyloxy)phenylpropionic acid: In vivo evaluation of antidiabetic activity / S. Kuranov, O. Luzina, M. Khvostov [et al.] // Pharmaceuticals. – 2020. – Vol. 13, No. 11. – P. 1-22. – DOI 10.3390/ph13110404. – EDN FQZBCN.
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Combined in silico, ex vivo, and in vivo assessment of L-17, a thiadiazine derivative with putative neuro-and cardioprotective and antidepressant effects / A. Sarapultsev, P. Sarapultsev, P. Vassiliev [et al.] // International Journal of Molecular Sciences. – 2021. – Vol. 22, No. 24. – P. 13626. – DOI 10.3390/ijms222413626. – EDN XXYYHM.
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Computational Analysis of CD46 Protein Interaction with SARS-CoV-2 Structural Proteins: Elucidating a Putative Viral Entry Mechanism into Human Cells / P. Vassiliev, E. Gusev, M. Komelkova [et al.] // Viruses. – 2023. – Vol. 15, No. 12. – P. 2297. – DOI 10.3390/v15122297. – EDN ZFWRSS.
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Consensus Ensemble Multitarget Neural Network Model of Anxiolytic Activity of Chemical Compounds and Its Use for Multitarget Pharmacophore Design / P. M. Vassiliev, D. V. Maltsev, A. A. Spasov [et al.] // Pharmaceuticals. – 2023. – Vol. 16, No. 5. – P. 731. – DOI 10.3390/ph16050731. – EDN BVBDWA.
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Hierarchical Assessment of the Structural Similarity of Pharmacologically Active Compounds / P. M. Vasil'ev, A. N. Kochetkov, L. R. Yanalieva [et al.] // Pharmaceutical Chemistry Journal. – 2021. – Vol. 54, No. 10. – P. 1019-1023. – DOI 10.1007/s11094-021-02314-2. – EDN DFBPMB.
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Neural network modeling search for multitarget RAGE inhibitors with different target activity spectra
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Searching for new anxiolytic agents among derivatives of 11-dialkylaminoethyl-2,3,4,5-tetrahydrodiazepino[1,2-a]benzimidazole / D. V. Maltsev, A. A. Spasov, D. S. Yakovlev [et al.] // European Journal of Pharmaceutical Sciences. – 2021. – Vol. 161. – P. 105792. – DOI 10.1016/j.ejps.2021.105792. – EDN KCDDUE.
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Synthesis and pharmacological evaluation of novel 2,3,4,5-tetrahydro[1,3]diazepino[1,2-a]benzimidazole derivatives as promising anxiolytic and analgesic agents / D. V. Maltsev, A. A. Spasov, P. M. Vassiliev [et al.] // Molecules. – 2021. – Vol. 26, No. 19. – P. 6049. – DOI 10.3390/molecules26196049. – EDN MGLYXM.
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