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2-Amino- and 2-hydroxymethylbenzimidazolium bromides as protein tyrosine phosphatase 1В (PTP1В) inhibitors and other targets associated with...
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2Е-бензилиден-19,28-эпоксиноролеананы: синтез и ингибирование α-глюкозидазы
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3-Arylidene-2-oxindoles as GSK3β inhibitors and anti-thrombotic agents / D. Babkov, E. Bezsonova, V. Sirotenko [et al.] // Bioorganic & Medicinal Chemistry Letters. – 2023. – Vol. 87. – P. 129283. – DOI 10.1016/j.bmcl.2023.129283. – EDN JLQKWC.
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3-Arylidene-2-oxindoles as Potent NRH:Quinone Oxidoreductase 2 Inhibitors / N. A. Lozinskaya, E. N. Bezsonova, M. Dubar [et al.] // Molecules. – 2023. – Vol. 28, No. 3. – P. 1174. – DOI 10.3390/molecules28031174. – EDN IQBSLQ.
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6-(Tetrazol-5-yl)-7-aminoazolo[1,5-a]pyrimidines as Novel Potent CK2 Inhibitors / G. V. Urakov, K. V. Savateev, S. K. Kotovskaya [et al.] // Molecules. – 2022. – Vol. 27, No. 24. – P. 8697. – DOI 10.3390/molecules27248697. – EDN JNFUYI.
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A Novel Dipterocarpol Derivative that Targets Alpha-Glucosidase and NLRP3 Inflammasome Activity for Treatment of Diabetes Mellitus / R. Danilov, I. E. Smirnova, Z. I. Galimova [et al.] // Chemistry & Biodiversity. – 2024. – DOI 10.1002/cbdv.202401626. – EDN HGOZNC.
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Amino Derivatives of Diaryl Pyrimidines and Azolopyrimidines as Protective Agents against LPS-Induced Acute Lung Injury / A. Spasov, I. Ovchinnikova, O. Fedorova [et al.] // Molecules. – 2023. – Vol. 28, No. 2. – P. 741. – DOI 10.3390/molecules28020741. – EDN APNGOY.
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Anti-Inflammatory Activity of Soluble Epoxide Hydrolase Inhibitors Based on Selenoureas Bearing an Adamantane Moiety / V. Burmistrov, Ch. Morisseau, D. A. Babkov [et al.] // International Journal of Molecular Sciences. – 2022. – Vol. 23, No. 18. – P. 10710. – DOI 10.3390/ijms231810710. – EDN VOZLJV.
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Azolo[5′,1′,2,3]pyrimido[5,4-e]tetrazolo[1,5-c]pyrimidines as dual-action antiglycators and α-glucosidase inhibitors
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